Iferanserin-hydrochloride-S-MPEC-hydrochloride-生命科学试剂-MCE.pdf

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Iferanserinhydrochloride

Cat.No.:HY-118557A

CASNo.:210350-29-1

Synonyms:S-MPEChydrochloride

分⼦式:C₂₃H₂₉ClN₂O

分⼦量:384.94

作⽤靶点:5-HTReceptor

作⽤通路:GPCR/GProtein;NeuronalSignaling

储存⽅式:Pleasestoretheproductundertherecommendedconditionsin

theCertificateofAnalysis.

BIOLOGICALACTIVITY

⽣物活性Iferanserinhydrochloride(S-MPEChydrochloride)是⼀种选择性⾎清素受体拮抗剂，具有抑制内部痔疮的潜

在作⽤。Iferanserinhydrochloride在进⾏的IIb期临床试验中显⽰出有效性和耐受性，能够显著减少患者报告

的出⾎和瘙痒症状。

REFERENCES

[1].HeroldA,etal.Intra-analIferanserin10mgBIDforhemorrhoiddisease:aprospective,randomized,double-blind,placebo-controlled

trial.ClinTher.2012Feb;34(2):329-40.

[2].Intra-analIferanserin10mgBIDforhemorrhoiddisease:aprospective,randomized,double-blind,placebo-controlledtrial

McePdfHeight

Caution:Producthasnotbeenfullyvalidatedformedicalapplications.

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